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Peptide & Hormone Therapies for Health, Performance & Longevity | Dr. Craig Koniver

In this episode, Dr. Craig Koniver, M.D., a board-certified physician trained at Brown University and Thomas Jefferson University, discusses the therapeutic application of peptides and hormones for enhancing physical and mental health and performance. We explore GLP-1 analogs for weight loss, BPC-157 for wound healing and reducing inflammation, as well as peptides that increase growth hormone, improve REM sleep, and enhance cognitive function. We also cover testosterone therapy, NAD, NMN, and NR supplementation, methylene blue for mitochondrial health, stem cell therapies, and supplements such as CoEnzyme Q10 and methylated B vitamins. Additionally, we discuss effective dosages, sourcing, safety considerations, and the importance of working with knowledgeable physicians. Whether you're currently using peptides or exogenous hormones, or simply curious about their potential benefits and risks, this episode provides the scientific rationale behind how peptides function, their potential to enhance mental and physical health, and how they can optimize performance. Access the full show notes for this episode: https://go.hubermanlab.com/Nya6k2f Pre-order Andrew's book, Protocols: https://go.hubermanlab.com/protocols Use Ask Huberman Lab, our chat-based tool, for summaries, clips, and insights from this episode: https://go.hubermanlab.com/tqqZoQT *Thank you to our sponsors* AG1: https://drinkag1.com/huberman Joovv: https://joovv.com/huberman BetterHelp: https://betterhelp.com/huberman Function: https://functionhealth.com/huberman Eight Sleep: https://eightsleep.com/huberman *Dr. Craig Koniver* Koniver Wellness: https://koniverwellness.com Koniver Aesthetics: https://koniveraesthetics.com Instagram: https://www.instagram.com/koniverwellness LinkedIn: https://www.linkedin.com/in/craig-koniver-md-4bb100126 *Timestamps* 00:00:00 Dr. Craig Koniver 00:04:52 Sponsors: Joovv & BetterHelp 00:07:40 What is a Peptide? 00:09:37 GLP-1 Agonists, Semaglutide Weight Loss, Brain Health 00:15:49 GLP-1 Microdoses, Muscle Loss; Inflammation 00:18:43 BPC-157, Inflammation 00:23:27 BPC-157, Injection & Oral Forms; Injury Repair 00:28:43 Sourcing, Anabolic Steroids, Testosterone 00:34:48 Black & Gray Market, Compounding Pharmacies, Purity 00:38:20 Sponsor: AG1 00:39:51 Partnering with a Physician, LPS 00:43:00 BPC-157, Pentadeca Arginate (PDA); Side Effects & Doses 00:46:35 Ipamorelin, GHRP-6, Sleep, Appetite; Tool: Sleep & Growth Hormone 00:54:17 Tesamorelin, Sermorelin, CJC-1295; Stacking Peptides 00:58:45 Sponsor: Function & Eight Sleep 01:01:54 Coenzyme Q10 (CoQ10), Mitochondrial Health 01:05:16 Prescriptions, Physicians & Trust 01:14:09 Agency in Your Health 01:17:13 MK-677, Appetite 01:19:32 Hexarelin; Growth Hormone Secretagogues Dosing 01:21:10 Methylated B Vitamins, Homocysteine 01:24:47 Peptides for Sleep, Pinealon, Epitalon 01:31:03 Glycine, Liver Detoxification; Dosage 01:37:19 GLP-1, Compounding Pharmacies 01:39:03 Stem Cell Therapy, PRP 01:41:18 Thymosin Alpha-1, Cerebrolysin & Brain Health 01:44:17 Peptides for Cognitive Function, Methylene Blue, Doses 01:50:20 Covid, NAD Infusion, NMN & NR Supplements 01:57:13 Nutritional Deficiencies; NAD Dose & Regimen, NMN & NR 02:07:53 PT-141, Vyleesi, Libido; Nausea 02:10:57 FDA Approval & Removal, Pharmaceutical Companies 02:20:17 Positivity, Mindset & Health 02:26:23 Zero-Cost Support, YouTube, Spotify & Apple Follow & Reviews, Sponsors, YouTube Feedback, Protocols Book, Social Media, Neural Network Newsletter #HubermanLab #Science #Health #Peptides #HormoneHealth #Longevity Disclaimer & Disclosures: https://www.hubermanlab.com/disclaimer

Andrew HubermanhostCraig Koniverguest
Oct 6, 20242h 29mWatch on YouTube ↗

At a glance

WHAT IT’S REALLY ABOUT

Peptides, NAD, and Mindset: Precision Tools For Modern Health Optimization

  1. Andrew Huberman interviews physician Dr. Craig Koniver about the emerging but rapidly expanding world of peptide and hormone-adjacent therapies for health, performance, and longevity. They explain what peptides are, how they differ from classic hormone replacement, and why many sit mechanistically between supplements and full-blown drugs. The discussion covers GLP‑1 agonists, BPC‑157 and its successor PDA, growth hormone secretagogues, pinealon for REM sleep, and NAD in both infusion and injectable forms, including real-world protocols and safety considerations.
  2. They also address serious sourcing issues—why compounding pharmacies and physician supervision are crucial compared to gray‑market “research chemical” vendors—and how recent FDA actions have sharply restricted many popular peptides. Beyond molecules, Koniver emphasizes that tools like peptides and NAD work best when layered on a foundation of sleep, exercise, nutrition, and especially a deliberately positive mindset, which he views as the most powerful long-term health lever.

IDEAS WORTH REMEMBERING

5 ideas

Use GLP‑1 agonists slowly and strategically to avoid muscle loss and rebound weight gain.

Koniver sees semaglutide and especially tirzepatide as powerful tools when used via microdosing from compounding pharmacies, starting very low and titrating slowly. He aims for ≤2 pounds of weight loss per week, combines them with resistance training and adequate protein, and often stacks with growth hormone secretagogues (e.g., tirzepatide + sermorelin) to preserve lean mass. Conventional high-dose protocols drive rapid loss, “Ozempic face,” and quick weight regain once stopped.

Avoid gray‑market peptides; work only with physicians using reputable compounding pharmacies.

Many online vendors label products “not for human consumption” and skip rigorous endotoxin and sterility testing. Koniver has seen anaphylaxis and serious inflammatory reactions from such products, largely driven by contaminants like LPS. FDA‑regulated compounding pharmacies must meet strict purity and sterility standards and allow customized dosing and stacking; his protocol always includes a physician consult, contraindication review, and careful dosing rather than self‑experimentation from the internet.

BPC‑157 is off the table, but PDA (Penta‑DCA arginate) is an emerging substitute for systemic repair.

BPC‑157 was one of Koniver’s most broadly useful peptides for systemic anti‑inflammatory effects and tendon/ligament repair, often injected subcutaneously away from the injury site with strong whole‑body benefits. After FDA removal, he now uses PDA—a single amino acid variant—with similar clinical outcomes so far. His starting dose: 250–500 mcg subcutaneously once daily, Monday–Friday, to support joint recovery, post‑viral inflammation, and general tissue healing.

Choose growth hormone secretagogues based on your specific goals: sleep and leanness vs. appetite and mass.

Ipamorelin (≈100 mcg at bedtime, 5 days on/2 off) is his “clean,” sleep‑supportive, fat‑loss‑favoring GH secretagogue with minimal side effects when dosed properly. Tesamorelin (≈2 mg) targets visceral fat and often works especially well in women. Hexarelin (≈100 mcg in the morning) is more of an energy/endurance enhancer. By contrast, GHRP‑6 and MK‑677 strongly stimulate appetite and may raise prolactin and cortisol; he reserves them for hard‑gainers who specifically want rapid muscle and strength gains.

Pinealon plus glycine can dramatically increase REM sleep and improve sleep architecture.

Pinealon is a very small pineal‑targeted peptide that, in Koniver’s practice and Huberman’s personal experience, can substantially increase REM sleep time and improve overall sleep quality without sedation or observed side effects. Koniver compounds pinealon with injectable glycine (for inhibitory neurotransmission and liver support) and typically doses it subcutaneously at bedtime. Huberman reports roughly doubling his REM sleep on nights he uses it and seeing better sleep even on off nights, consistent with pineal support rather than simple sedation.

WORDS WORTH SAVING

5 quotes

Most of the medicines prescribed, particularly in America, are prescribed off label, meaning they've never ever been approved for what they're used.

Dr. Craig Koniver

If I can help people lose weight first, literally by using something like tirzepatide, then they're going to be motivated. The light bulb turns on, and that's the aha moment that I love helping people with.

Dr. Craig Koniver

Anything you expose yourself to continually doesn't work as well.

Dr. Craig Koniver

If I had to pick one thing for people, engaging in NAD would be it.

Dr. Craig Koniver

No good has ever come from a negative thought.

Dr. Craig Koniver

Basics of peptides and how they differ from hormones and supplementsGLP‑1 agonists (semaglutide, tirzepatide): microdosing, muscle loss, and metabolic effectsBPC‑157, FDA removal, and PDA (Penta‑DCA arginate) as a successorGrowth hormone secretagogues (ipamorelin, tesamorelin, GHRP‑6, hexarelin, MK‑677) for sleep, fat loss, and recoveryNAD (IV, subcutaneous, NMN/NR) for mitochondrial function, fatigue, and moodSleep‑specific peptides: pinealon plus glycine, REM sleep, and circadian supportRegulation, FDA crackdowns, compounding pharmacies vs. gray/black market, and the role of mindset in health

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